SCHEMBL30401740

SCHEMBL30401740

COc1ccc(-c2cc3c(N)c(C)ccc3c(N)n2)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.50
KDM4E B2RXH2 7/20 0.46
ALDH1A1 P00352 5/20 0.46
MAPT P10636 4/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
GFER P55789 1/20 0.46
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
RAD52 P43351 1/20 0.45
ACACA Q13085 1/20 0.45
ATM Q13315 2/20 0.45
USP2 O75604 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25372907 1.00 DHFR (0.50) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL25374933 0.88 KMO (0.42) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL30401294 0.88 KMO (0.42) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL509108 0.84 ACACA (0.51) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL25377685 0.83 SYK (0.54) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL30402644 0.83 SYK (0.54) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL509771 0.80 KDM4E (0.52) DHFRKDM4EALDH1A1MAPTMEN1
SCHEMBL25377291 0.79 PIK3CA (0.46) MAPT
SCHEMBL30402496 0.79 PIK3CA (0.46) MAPT
SCHEMBL15068737 0.77 KDM4E (0.42) KDM4EALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096718-A Aryl amide compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-05-09 CN disclosed