SCHEMBL304038

SCHEMBL304038

Cn1nccc1S(=O)(=O)N(Cc1ccc(Cl)cc1)c1cccc(N2CCCC2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
CNR2 P34972 2/20 0.41
KMT2A Q03164 1/20 0.40
LMNA P02545 3/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39
HTR2C P28335 2/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
DRD3 P35462 1/20 0.38
HTR6 P50406 1/20 0.38
HCRTR1 O43613 1/20 0.37
PKM P14618 1/20 0.37
MAPT P10636 1/20 0.36
PARP1 P09874 2/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL302085 0.83 CNR2 (0.47) NPC1CNR2LMNAPOLBHTT
SCHEMBL304739 0.78 CNR2 (0.43) NPC1RAB9ACNR2KMT2ALMNA
SCHEMBL3275899 0.76 HTR2C (0.49) NPC1RAB9ACNR2LMNAALDH1A1
SCHEMBL2188016 0.74 KDM4E (0.43) NPC1KMT2ALMNAPOLBALDH1A1
SCHEMBL3275051 0.74 HTR2C (0.45) NPC1RAB9ACNR2KMT2AALDH1A1
SCHEMBL301863 0.73 MEN1 (0.49) NPC1RAB9AKMT2AALDH1A1
SCHEMBL302155 0.73 MEN1 (0.47) NPC1RAB9AKMT2AALDH1A1
SCHEMBL1971605 0.72 CNR2 (0.38) NPC1RAB9ACNR2KMT2ALMNA
SCHEMBL3260086 0.72 TSHR (0.39) NPC1RAB9ACNR2KMT2ALMNA
SCHEMBL1976194 0.71 CNR2 (0.39) NPC1RAB9ACNR2KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500835-A 2012-01-12 JP claimed
EP-2334637-A1 NOVEL POTASSIUM CHANNEL BLOCKERS Xention Limited (GB) 2011-06-22 EP claimed
EP-2334637-A1 NOVEL POTASSIUM CHANNEL BLOCKERS Xention Limited (GB) 2011-06-22 EP disclosed