SCHEMBL3041969

SCHEMBL3041969

O=C(OC(CCc1ccccc1)NCc1ccc(-c2ccc3[nH]cnc3c2)cc1)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 10/20 0.37
IP6K1 Q92551 2/20 0.35
IP6K3 Q96PC2 1/20 0.35
IP6K2 Q9UHH9 1/20 0.35
NAMPT P43490 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRA6 Q16445 1/20 0.34
QPCTL Q9NXS2 2/20 0.33
MME P08473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MMP12 P39900 2/20 0.32
S1PR1 P21453 1/20 0.32
BCHE P06276 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3047194 0.84 HTT (0.35) QPCTNAMPTALDH1A1
SCHEMBL3037465 0.84 POLB (0.33) QPCT
SCHEMBL3051555 0.84 QPCT (0.38) QPCTNAMPTMME
SCHEMBL3034900 0.83 TEK (0.43) MME
SCHEMBL3051311 0.83 QPCT (0.37) QPCT
SCHEMBL3038470 0.82 EPHB4 (0.35)
SCHEMBL3049024 0.79 LMNA (0.41) QPCT
SCHEMBL3044920 0.79 MTOR (0.36) NAMPT
Trifluoroacetic Acid SCHEMBL3041965 0.77 HDAC1 (0.47) BCHE
SCHEMBL3823826 0.74 MAOB (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 QPCT 1796/4885IP6K1 1533/4885IP6K3 1510/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.