SCHEMBL30433593

SCHEMBL30433593

O=c1ccc2ccc(-c3ccncc3)cc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 10/20 0.59
PDE3A Q14432 10/20 0.59
CYP19A1 P11511 1/20 0.47
AAK1 Q2M2I8 2/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA3 P07451 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
CLK1 P49759 1/20 0.45
MGLL Q99685 1/20 0.44
GSK3B P49841 1/20 0.44
MAPK1 P28482 1/20 0.44
PDPK1 O15530 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4287747 0.88 PDE3B (0.57) PDE3BPDE3ACYP19A1CA12CA1
SCHEMBL27805572 0.81 CA12 (0.59) PDE3BPDE3ACA12CA1CA3
SCHEMBL17067225 0.80 FGFR1 (0.59) PDE3BPDE3ACYP19A1
SCHEMBL23207309 0.76 CA9 (0.62) PDE3BPDE3ACA12CA1CA3
SCHEMBL18000095 0.75 PDE3B (0.50) PDE3BPDE3AAAK1CLK1PDPK1
SCHEMBL4553604 0.75 CDK5 (0.46) CA12CA1CA3CA4CA6
SCHEMBL9599136 0.74 ALDH1A1 (0.57) PDE3BPDE3AGSK3BMAPK1
SCHEMBL18000228 0.74 BRAF (0.58) PDE3BPDE3ACLK1PDPK1
SCHEMBL31192609 0.74 PDE3B (1.00) PDE3BPDE3ACLK1PDPK1
SCHEMBL20494235 0.73 KDM4E (0.51) PDE3BPDE3APDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081212-A1 METHODS OF USING ALK2 INHIBITORS KEROS THERAPEUTICS, INC. (US) 2023-05-11 WO disclosed