SCHEMBL9599136

SCHEMBL9599136

O=c1ccc2cc3nc(-c4ccncc4)[nH]c3cc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
KDM4E B2RXH2 4/20 0.57
HPGD P15428 4/20 0.57
HSD17B10 Q99714 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
RHEB Q15382 1/20 0.57
NPC1 O15118 3/20 0.52
RAB9A P51151 2/20 0.52
PKN1 Q16512 5/20 0.52
PKN2 Q16513 5/20 0.52
PDE3B Q13370 2/20 0.52
PDE3A Q14432 2/20 0.52
PDE4A P27815 1/20 0.52
PDE4B Q07343 1/20 0.52
PDE4C Q08493 1/20 0.52
PDE4D Q08499 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9598691 0.83 MAPT (0.68) ALDH1A1KDM4EHPGDHSD17B10NPC1
SCHEMBL9598512 0.81 PRKD3 (0.43) ALDH1A1KDM4ERHEBNPC1RAB9A
SCHEMBL9599277 0.81 SLC2A1 (0.55) ALDH1A1KDM4EHPGDHSD17B10NPC1
SCHEMBL9598976 0.80 FBP1 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9678498 0.80 ALDH1A1 (0.62) ALDH1A1KDM4EHPGDHSD17B10CYP1A2
SCHEMBL9378150 0.80 ALDH1A1 (0.62) ALDH1A1KDM4EHPGDHSD17B10CYP1A2
SCHEMBL9379605 0.79 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDHSD17B10CYP1A2
SCHEMBL9704460 0.75 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDHSD17B10CYP1A2
SCHEMBL30433593 0.74 PDE3B (0.59) PDE3BPDE3AGSK3BMAPK1
SCHEMBL9679051 0.74 PDE3B (0.57) ALDH1A1KDM4EHPGDHSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5212186-A Asthma, anticoagulant BEIERSDORF AKTIENGESELLSCHAFT (DE) 1993-05-18 US disclosed
EP-0473963-A1 Pyrrolobenzimidazoles, imidazobenzoxazinones, and imidazoquinolones, processes for their preparation and their use as well as compositions containing these compounds Beiersdorf-Lilly GmbH (DE) 1992-03-11 EP disclosed