SCHEMBL30438783

SCHEMBL30438783

Cn1c(=O)c2[nH]c(-c3cc4ccccc4n3C)nc2n(C)c1=O

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.64
ADORA2B P29275 2/20 0.64
CYP1A2 P05177 1/20 0.64
ADORA3 P0DMS8 1/20 0.64
ADORA2A P29274 1/20 0.64
ADORA1 P30542 1/20 0.64
BLM P54132 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
HSD17B10 Q99714 1/20 0.64
ALDH1A1 P00352 1/20 0.58
HPGD P15428 1/20 0.58
TDP1 Q9NUW8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28527789 0.82 ADORA2B (0.63) KDM4EADORA2BCYP1A2ADORA3ADORA2A
8-Phenyl Theophylline SCHEMBL516432 0.78 ADORA2A (1.00) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL25090657 0.78 ADORA2B (0.73) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL28909317 0.76 KDM4E (0.62) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL30438203 0.76 KDM4E (0.62) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL8596143 0.76 KDM4E (0.76) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL29429838 0.75 KDM4E (0.70) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL516349 0.75 KDM4E (0.70) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL25090354 0.74 KDM4E (0.72) KDM4EADORA2BCYP1A2ADORA3ADORA2A
SCHEMBL2119734 0.74 KDM4E (0.72) KDM4EADORA2BCYP1A2ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112209930-B Itratheophylline derivative, and preparation method and application thereof 山东新华制药股份有限公司 2023-05-16 CN disclosed