SCHEMBL30440463

SCHEMBL30440463

COc1ccc(Oc2cnc(C#N)cc2OC)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.49
GAA P10253 2/20 0.49
AR P10275 2/20 0.48
MAP2K1 Q02750 2/20 0.44
MAPK1 P28482 2/20 0.42
TSHR P16473 1/20 0.42
PDE10A Q9Y233 1/20 0.42
FGFR2 P21802 1/20 0.42
CSF1R P07333 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGDS O60760 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
NQO1 P15559 1/20 0.41
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21045734 1.00 POLB (0.49) POLBGAAARMAP2K1MAPK1
SCHEMBL21081168 0.91 AR (0.60) POLBGAAARMAP2K1MAPK1
SCHEMBL21045893 0.91 MAP2K1 (0.49) POLBGAAARMAP2K1MAPK1
SCHEMBL21045605 0.89 L3MBTL1 (0.53) POLBARMAP2K1MAPK1PDE10A
SCHEMBL21045783 0.89 CYP1A2 (0.47) POLBGAAARPDGFRASLC22A12
SCHEMBL21045778 0.87 TRPC6 (0.44) POLBGAAARMAP2K1MAPK1
SCHEMBL21045809 0.86 TRPC6 (0.44) POLBGAAARMAP2K1MAPK1
SCHEMBL21045646 0.86 RAB9A (0.45) ARTSHRFGFR2ALDH1A1L3MBTL1
SCHEMBL21045704 0.86 AR (0.42) POLBGAAARMAP2K1PDE10A
SCHEMBL30439308 0.86 RAB9A (0.45) ARTSHRFGFR2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111527078-B Pyridinecarbonyl derivatives and their therapeutic use as TRPC6 inhibitors 勃林格殷格翰国际公司 2023-06-02 CN disclosed