SCHEMBL30449529

SCHEMBL30449529

Cc1cccc(-n2nc(C(=O)O)cc2-c2ccc3ncsc3c2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 7/20 0.46
RPA1 P27694 3/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MDM2 Q00987 3/20 0.41
MCL1 Q07820 3/20 0.41
BCL2 P10415 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HKDC1 Q2TB90 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MARS1 P56192 1/20 0.40
PPP1CA P62136 2/20 0.39
ACVR1B P36896 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20955450 1.00 TGFBR1 (0.46) TGFBR1RPA1KDM4EALDH1A1MDM2
SCHEMBL20955667 0.91 TGFBR1 (0.47) TGFBR1MARS1ACVR1B
SCHEMBL20979040 0.88 PFKFB3 (0.45) TGFBR1KDM4EALDH1A1NPC1RAB9A
SCHEMBL20955280 0.88 TGFBR1 (0.44) TGFBR1ALDH1A1MDM2MCL1BCL2
SCHEMBL25336136 0.86 TGFBR1 (0.45) TGFBR1ACVR1B
SCHEMBL20978891 0.86 TGFBR1 (0.57) TGFBR1ACVR1B
SCHEMBL21129341 0.86 CACNA1G (0.49) TGFBR1RPA1KDM4EALDH1A1
SCHEMBL29425326 0.85 TGFBR1 (0.44) TGFBR1KDM4ENPC1RAB9AHKDC1
SCHEMBL25335613 0.85 TGFBR1 (0.44) TGFBR1KDM4ENPC1RAB9AHKDC1
SCHEMBL20979169 0.85 PFKFB3 (0.46) TGFBR1KDM4EALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116249692-B Pyrazole compound as well as preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-08-23 CN disclosed
CN-116249692-A Pyrazole compound as well as preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-06-09 CN disclosed