SCHEMBL30451265

SCHEMBL30451265

Cc1ccccc1C1NC(=O)c2c(C)cccc21

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.56
HTR2A P28223 4/20 0.56
HTR2B P41595 4/20 0.56
PBRM1 Q86U86 5/20 0.50
TNKS2 Q9H2K2 2/20 0.46
ALDH1A1 P00352 4/20 0.44
GSK3B P49841 1/20 0.43
BACE1 P56817 1/20 0.43
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30451575 0.85 AURKA (0.44) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL29016841 0.80 PBRM1 (0.60) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL12716352 0.78 HTR2A (0.55) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL11358726 0.76 HTR2A (0.54) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL29010215 0.74 HTR2A (0.51) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL12718314 0.74 HTR2A (0.51) HTR2CHTR2AHTR2BPBRM1TNKS2
SCHEMBL13756918 0.72 HTR2A (1.00) HTR2CHTR2AHTR2B
SCHEMBL13756919 0.72 HTR2A (1.00) HTR2CHTR2AHTR2B
SCHEMBL30451582 0.71 TNKS2 (0.47) HTR2CHTR2AHTR2BPBRM1TNKS2
Hydrochloric Acid SCHEMBL4467236 0.71 HTR2A (1.00) HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed