SCHEMBL30452455

SCHEMBL30452455

CCS(=O)(=O)c1ccc(CBr)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.37
PSIP1 O75475 2/20 0.35
RIPK1 Q13546 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTR6 P50406 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
DDR1 Q08345 1/20 0.32
KDM2B Q8NHM5 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
KCNA5 P22460 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20300406 1.00 CA2 (0.37) CA2PSIP1RIPK1CYP1A2CYP2D6
SCHEMBL1940002 0.84 CCR2 (0.40)
SCHEMBL30457289 0.84 CCR2 (0.40)
SCHEMBL20300285 0.82 CA2 (0.44) CA2PSIP1RIPK1CYP4F2CYP4A11
SCHEMBL24050785 0.80 CA2 (0.41) CA2
SCHEMBL24050330 0.80 TRPV4 (0.36) CA2CYP4F2CYP4A11KCNA5
SCHEMBL14744537 0.78 HPGD (0.43) CA2KMT2ATDP1TSHR
SCHEMBL16011120 0.78 NMT1 (0.47) CA2TDP1DDR1TSHR
SCHEMBL776801 0.77 AKR1B1 (0.44) CA2HTR6DDR1KDM2BTSHR
SCHEMBL1795036 0.77 USP30 (0.39) CYP2C9KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116162084-A Pyran derivatives as CYP11A1 inhibitors 奥赖恩公司 2023-05-26 CN disclosed