SCHEMBL30453395

SCHEMBL30453395

Nc1ncc(-c2cccc(C(=O)NCCN3CCOCC3)c2)nc1OCc1c(F)ccc(F)c1Cl

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.54
ATR Q13535 2/20 0.50
GRK5 P34947 1/20 0.49
PIK3CD O00329 1/20 0.49
PIK3CG P48736 1/20 0.49
ABL1 P00519 1/20 0.48
BCR P11274 1/20 0.48
EPHX2 P34913 1/20 0.46
CAMK2D Q13557 1/20 0.46
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ERN1 O75460 1/20 0.45
HPGDS O60760 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTR1A P08908 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
KCNH2 Q12809 1/20 0.44
CD274 Q9NZQ7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488692 1.00 MAP4K4 (0.54) MAP4K4ATRGRK5PIK3CDPIK3CG
SCHEMBL30452963 0.96 MAP4K4 (0.49) MAP4K4ATRGRK5PIK3CDPIK3CG
SCHEMBL488205 0.96 MAP4K4 (0.49) MAP4K4ATRGRK5PIK3CDPIK3CG
SCHEMBL488217 0.93 ATR (0.58) MAP4K4ATRCAMK2DERN1
SCHEMBL30454379 0.93 ATR (0.58) MAP4K4ATRCAMK2DERN1
SCHEMBL488479 0.92 CD274 (0.50) MAP4K4ATREPHX2HPGDSALDH1A1
SCHEMBL30453023 0.92 CD274 (0.50) MAP4K4ATREPHX2HPGDSALDH1A1
SCHEMBL487865 0.90 ATR (0.49) MAP4K4ATRGRK5
SCHEMBL488105 0.89 ATR (0.53) MAP4K4ATR
SCHEMBL30453359 0.89 ATR (0.53) MAP4K4ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed