SCHEMBL30455313

SCHEMBL30455313

COc1cc(-c2ccc3nc(C)[nH]c(=O)c3c2)ccc1Cc1nccs1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.47
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 1/20 0.46
ACVR1 Q04771 2/20 0.44
ROCK2 O75116 1/20 0.41
GUSB P08236 1/20 0.40
POLB P06746 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP1B1 Q16678 1/20 0.38
CASR P41180 1/20 0.37
IP6K1 Q92551 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29002513 1.00 TRPV1 (0.47) TRPV1KDM4EHSD17B10LMNAACVR1
SCHEMBL29002558 0.80 CASR (0.38) MEN1KMT2ACASR
SCHEMBL30454826 0.77 HSD17B10 (0.49) TRPV1KDM4EHSD17B10LMNAACVR1
SCHEMBL30454449 0.71 KDM4E (0.49) TRPV1KDM4EHSD17B10LMNAACVR1
Ammonia Solution, Strong SCHEMBL3162475 0.69 APLNR (0.50) KDM4ELMNAMEN1KMT2ACYP1A2
SCHEMBL29002566 0.69 PYCR1 (0.41) KDM4ELMNAPOLBALDH1A1MAPT
SCHEMBL30455640 0.67 KDM4E (0.46) TRPV1KDM4EHSD17B10LMNAACVR1
SCHEMBL29002511 0.67 KDM4E (0.46) TRPV1KDM4EHSD17B10LMNAACVR1
SCHEMBL1257374 0.65 KDM4E (1.00) TRPV1KDM4EHSD17B10LMNAGUSB
SCHEMBL29900577 0.65 KDM4E (1.00) TRPV1KDM4EHSD17B10LMNAGUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143708-A Polysubstituted benzazepine heteroaryl derivative and application thereof 四川汇宇制药股份有限公司 2023-05-23 CN disclosed