SCHEMBL30457513

SCHEMBL30457513

CC(C)(C)OC(=O)NCc1ccc(F)c(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.47
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
IDO1 P14902 1/20 0.44
NAMPT P43490 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
KDM4A O75164 1/20 0.43
AAK1 Q2M2I8 1/20 0.43
HDAC1 Q13547 1/20 0.42
TSHR P16473 1/20 0.42
FPR3 P25089 1/20 0.42
FPR2 P25090 1/20 0.42
GLS O94925 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL51488 1.00 GRM2 (0.47) GRM2GAAL3MBTL1IDO1NAMPT
SCHEMBL507617 0.89 GRM2 (0.47) GRM2GAAL3MBTL1NAMPTCA1
SCHEMBL24999627 0.87 GRM2 (0.49) GRM2GAAL3MBTL1NAMPTKDM4A
SCHEMBL29769069 0.87 GRM2 (0.49) GRM2GAAL3MBTL1NAMPTKDM4A
SCHEMBL17823099 0.86 CA2 (0.49) IDO1NAMPTCA1CA2AAK1
SCHEMBL31142951 0.86 ALDH1A1 (0.48) GRM2GAAL3MBTL1NAMPTCA1
SCHEMBL3688009 0.84 HDAC1 (0.48) GRM2GAAL3MBTL1NAMPTCA1
SCHEMBL1985433 0.84 HDAC1 (0.51) GRM2GAAL3MBTL1NAMPTCA1
SCHEMBL16020300 0.84 MMP13 (0.54) GRM2GAAL3MBTL1NAMPTKDM4A
SCHEMBL31142856 0.84 NOTUM (0.48) GRM2GAAL3MBTL1NAMPTCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4448508-A1 BENZOTHIOPHENE DERIVATIVES AS RXFP1 AGONISTS Bristol-Myers Squibb Company (US) 2024-10-23 EP disclosed
WO-2023114823-A1 BENZOTHIOPHENE DERIVATIVES AS RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed