SCHEMBL30458103

SCHEMBL30458103

CC1(NCc2ccc(C(F)(F)F)c(Br)c2)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.45
EPHX2 P34913 1/20 0.42
GPR119 Q8TDV5 1/20 0.41
HDAC1 Q13547 3/20 0.39
HDAC2 Q92769 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MEN1 O00255 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NAMPT P43490 2/20 0.39
CYP2C9 P11712 1/20 0.39
ANO1 Q5XXA6 1/20 0.38
PKM P14618 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 2/20 0.38
NOTUM Q6P988 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20570228 1.00 TACR1 (0.45) TACR1EPHX2GPR119HDAC1HDAC2
SCHEMBL30458402 0.81 TACR1 (0.42) TACR1EPHX2GPR119HDAC1HDAC8
SCHEMBL20569877 0.81 TACR1 (0.42) TACR1EPHX2GPR119HDAC1HDAC8
SCHEMBL14279760 0.81 ANO1 (0.47) TACR1GPR119HDAC1HDAC2SMN1; SMN2
SCHEMBL20766101 0.81 HDAC2 (0.51) TACR1HDAC1HDAC2SMN1; SMN2MEN1
SCHEMBL3658891 0.80 SMN1; SMN2 (0.46) TACR1HDAC1HDAC2SMN1; SMN2MEN1
SCHEMBL20566981 0.80 TACR1 (0.47) TACR1EPHX2GPR119HDAC1HDAC2
SCHEMBL18064777 0.79 IDO1 (0.46) CYP2C19CYP2C9
SCHEMBL3661148 0.79 GPR119 (0.44) TACR1GPR119NAMPT
SCHEMBL2798269 0.78 KEAP1 (0.44) GPR119MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678177-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-06-13 CN disclosed