SCHEMBL30458402

SCHEMBL30458402

CN(Cc1ccc(C(F)(F)F)c(Br)c1)C1(C)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.42
GPR119 Q8TDV5 5/20 0.40
EPHX2 P34913 1/20 0.40
MGLL Q99685 1/20 0.39
PKM P14618 1/20 0.38
RORC P51449 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20569877 1.00 TACR1 (0.42) TACR1GPR119EPHX2MGLLPKM
SCHEMBL20571126 0.86 GPR119 (0.41) TACR1GPR119EPHX2MGLL
SCHEMBL20570228 0.81 TACR1 (0.45) TACR1GPR119EPHX2PKMHDAC1
SCHEMBL30458103 0.81 TACR1 (0.45) TACR1GPR119EPHX2PKMHDAC1
SCHEMBL20567721 0.80 MGLL (0.50) TACR1GPR119EPHX2MGLLPKM
SCHEMBL18064777 0.78 IDO1 (0.46) MGLL
SCHEMBL25487285 0.77 GPR119 (0.41) TACR1GPR119EPHX2MGLLPKM
SCHEMBL20570689 0.74 FFAR4 (0.41) MGLL
SCHEMBL20571082 0.73 MGLL (0.40) MGLL
SCHEMBL20567325 0.73 MGLL (0.57) TACR1GPR119MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678177-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-06-13 CN disclosed