SCHEMBL30465799

SCHEMBL30465799

Cc1ccc2c(c1)C(=O)CC2

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.59
PARP10 Q53GL7 2/20 0.56
PARP1 P09874 1/20 0.56
BRD4 O60885 2/20 0.49
METAP1 P53582 2/20 0.48
ACHE P22303 1/20 0.48
TYMS P04818 2/20 0.46
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
CYP19A1 P11511 2/20 0.45
CYP11B2 P19099 2/20 0.45
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP11 Q9NR21 1/20 0.43
PTGS2 P35354 1/20 0.42
ELANE P08246 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL354988 1.00 PBRM1 (0.59) PBRM1PARP10PARP1BRD4METAP1
SCHEMBL21234894 0.88 METAP1 (0.55) PBRM1PARP10PARP1BRD4METAP1
SCHEMBL29673118 0.88 MAOA (0.59) PBRM1PARP10PARP1METAP1ACHE
SCHEMBL1274936 0.88 MAOA (0.59) PBRM1PARP10PARP1METAP1ACHE
SCHEMBL10177012 0.88 MAOA (0.59) PBRM1PARP10PARP1METAP1ACHE
SCHEMBL14925847 0.84 METAP1 (0.60) PARP10PARP1METAP1ACHETYMS
SCHEMBL5208267 0.84 BRD4 (0.55) PBRM1PARP10PARP1BRD4TYMS
SCHEMBL5929505 0.83 CYP2A6 (0.58) PBRM1PARP10PARP1BRD4METAP1
SCHEMBL29726014 0.83 CASP1 (0.59) PBRM1PARP10PARP1METAP1MAOA
SCHEMBL423287 0.83 CASP1 (0.59) PBRM1PARP10PARP1METAP1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116940552-A Spirocyclic hexane derivatives, pharmaceutical compositions containing them and their use as anti-apoptotic inhibitors 法国施维雅药厂 2023-10-24 CN disclosed
WO-2023122754-A1 PROCESSES AND INTERMEDIATES FOR PREPARING GB13, GB22 AND HIMGALINE THE SCRIPPS RESEARCH INSTITUTE (US) 2023-06-29 WO disclosed