SCHEMBL3046785

SCHEMBL3046785

Fc1cc(-c2ccc3[nH]cnc3c2)ccc1CNC1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PABPC1 P11940 1/20 0.41
HTT P42858 4/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39
EPHX1 P07099 1/20 0.38
ALDH1A1 P00352 2/20 0.37
ALOX15 P16050 2/20 0.37
PARP1 P09874 1/20 0.37
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
BACE1 P56817 1/20 0.35
IP6K1 Q92551 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13137099 1.00 PABPC1 (0.41) PABPC1HTTLMNAKMT2AHRH3
SCHEMBL3043972 0.87 BACE1 (0.37) BCHEACHEBACE1CXCR3QPCT
Hydrochloric Acid SCHEMBL3034125 0.86 BACE1 (0.36) BCHEACHEBACE1CXCR3QPCT
SCHEMBL13137108 0.85 QPCT (0.34) BCHEACHEBACE1QPCTQPCTL
SCHEMBL3041921 0.84 OPRM1 (0.38) BCHEACHEBACE1QPCTQPCTL
SCHEMBL13137097 0.84 HDAC3 (0.45) KMT2AEPHX1MEN1CXCR3QPCT
Hydrochloric Acid SCHEMBL3047516 0.84 QPCT (0.33) BCHEACHEBACE1QPCTQPCTL
Hydrochloric Acid SCHEMBL3040445 0.84 OPRM1 (0.37) BCHEACHEBACE1QPCTQPCTL
Hydrochloric Acid SCHEMBL3037830 0.84 HDAC3 (0.44) KMT2AEPHX1MEN1CXCR3QPCT
SCHEMBL13137098 0.83 BCHE (0.36) KMT2AEPHX1BCHEMEN1QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US claimed
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 PABPC1 3642/4885HTT 1472/4885LMNA 4551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.