SCHEMBL30480858

SCHEMBL30480858

CCc1cc2c(Br)cccc2[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.54
DDO Q99489 2/20 0.54
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 3/20 0.42
HRH4 Q9H3N8 1/20 0.42
HTT P42858 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
HSD17B10 Q99714 3/20 0.40
NPEPPS P55786 1/20 0.40
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627652 0.80 KDM4E (0.45) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL22571313 0.80 DAO (0.61) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL29471220 0.79 BRD4 (0.53) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL26551030 0.79 BRD4 (0.53) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL23714709 0.77 PARP1 (0.42) DAODDOKDM4EALDH1A1HRH4
SCHEMBL15690473 0.76 DAO (0.65) DAODDOKDM4EALDH1A1HRH4
SCHEMBL15690324 0.75 GRIN2D (0.51) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL25203298 0.74 KDM4E (0.56) RAB9AKDM4EALDH1A1PDE3BPDE3A
SCHEMBL12277902 0.72 MEN1 (0.62) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL31154599 0.72 KDM4E (0.66) DAODDOKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116368128-A Heterocyclic compounds as CBP/EP300 bromodomain inhibitors 奥瑞基尼肿瘤有限公司 2023-06-30 CN disclosed