SCHEMBL30484457

SCHEMBL30484457

Fc1ccc(-c2ccc(-c3ccnc(CN4CCC5(CCCC5)CC4)c3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.50
HTR1A P08908 1/20 0.50
DRD4 P21917 5/20 0.42
DRD3 P35462 5/20 0.42
SSTR5 P35346 1/20 0.38
KCNH2 Q12809 1/20 0.38
CXCR4 P61073 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
ACKR3 P25106 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GFER P55789 1/20 0.36
CSNK1D P48730 1/20 0.36
CSNK1E P49674 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30484462 0.88 EGLN1 (0.47) DRD2HTR1AEGLN1KDM4EALDH1A1
SCHEMBL30484482 0.87 EGLN1 (0.46) DRD2HTR1AEGLN1KDM4EALDH1A1
SCHEMBL30484425 0.87 HTR1A (0.39) DRD2HTR1ACXCR4EGLN1KDM4E
SCHEMBL30484511 0.87 LSS (0.46) DRD2HTR1ADRD4DRD3CXCR4
SCHEMBL30484434 0.84 SIGMAR1 (0.41) DRD2HTR1AKCNH2CXCR4EGLN1
SCHEMBL10373480 0.82 SSTR5 (0.49) DRD2HTR1ADRD4DRD3SSTR5
SCHEMBL10372410 0.80 OPRL1 (0.50) DRD2HTR1ADRD4DRD3SSTR5
SCHEMBL30484486 0.79 EGLN1 (0.40) DRD2HTR1AEGLN1KDM4EALDH1A1
SCHEMBL30484426 0.79 TMEM97 (0.40) DRD2HTR1AKCNH2CXCR4EGLN1
SCHEMBL27425923 0.78 DRD2 (0.51) DRD2HTR1ADRD4DRD3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116354897-B Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2024-10-15 CN disclosed
CN-116354897-A Substituted 1,2, 4-triazole, pyridine and pyrimidine derivatives and application thereof in medicines 华东师范大学 2023-06-30 CN disclosed