SCHEMBL30487378

SCHEMBL30487378

CC(C)(C)OC(=O)N1Cc2ccc(F)cc2C(CO)C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.44
NR1H2 P55055 2/20 0.43
NAMPT P43490 1/20 0.42
DPP8 Q6V1X1 3/20 0.41
DPP9 Q86TI2 3/20 0.41
HPGDS O60760 1/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 1/20 0.39
DPP4 P27487 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
BRD3 Q15059 2/20 0.39
MAPK1 P28482 1/20 0.38
TAOK3 Q9H2K8 1/20 0.38
TACR1 P25103 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25290544 1.00 ESR2 (0.44) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL30487414 0.88 NAMPT (0.45) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL25251748 0.88 NAMPT (0.45) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL25251450 0.84 ESR2 (0.44) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL30487370 0.84 ESR2 (0.44) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL14101075 0.80 TGFBR1 (0.42) ESR2NR1H2NAMPTDPP7GPR119
SCHEMBL13337056 0.77 DPP9 (0.58) ESR2NR1H2NAMPTDPP8DPP9
SCHEMBL22366343 0.74 NAMPT (0.52) ESR2NR1H2NAMPTGPR119DDB1
SCHEMBL30428022 0.74 NAMPT (0.52) ESR2NR1H2NAMPTGPR119DDB1
SCHEMBL31067462 0.73 ESR2 (0.74) ESR2NR1H2NAMPTDPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125935-A1 BENZOPYRIDINE DERIVATIVE REGULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2023-07-06 WO disclosed