SCHEMBL30487482

SCHEMBL30487482

COC(=O)C[C@H](NC(=O)C1CC2(C1)CN(CCCC(C)=O)C2)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.34
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
WDR5 P61964 1/20 0.32
HDAC3 O15379 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC8 Q9BY41 1/20 0.32
ITGB1 P05556 2/20 0.31
ITGA4 P13612 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21314515 0.91 ITGB1 (0.38) HDAC1ITGB3ITGA2BITGB1ITGA4
SCHEMBL20157749 0.86 HDAC1 (0.41) HDAC1ITGB3ITGA2B
SCHEMBL20141286 0.82 ITGB1 (0.35) ITGB3ITGA2BWDR5ITGB1ITGA4
SCHEMBL30487546 0.82 SUCNR1 (0.40) HDAC1ITGB3WDR5HDAC3HDAC2
SCHEMBL26462366 0.79 ITGB3 (0.35) ITGB3ITGA2BWDR5ITGB1ITGA4
SCHEMBL30487506 0.79 ITGAV (0.55) ITGB3ITGA2BITGB1
SCHEMBL21317534 0.79 ITGAV (0.55) ITGB3ITGA2BITGB1
SCHEMBL21317519 0.79 STS (0.41) ITGB3ITGA2BITGB1ITGA4
SCHEMBL21314447 0.77 WDR5 (0.34) HDAC1ITGB3ITGA2BWDR5HDAC3
SCHEMBL21314446 0.77 WDR5 (0.34) HDAC1ITGB3ITGA2BWDR5HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11639353-B2 Cyclobutanes- and azetidine-containing mono and spirocyclic compounds as αV integrin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2023-05-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11639353-B2 Cyclobutanes- and azetidine-containing mono and spirocyclic compounds as αV integrin inhibitors ITGB1, ITGB2, ITGA1 HDAC1 420/4885ITGB3 6/4885ITGA2B 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.