SCHEMBL30508296

SCHEMBL30508296

O=C(O)c1ccc(-c2cnn3cc(-c4ccc(N5CCOCC5)cc4)cnc23)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.66
PRKAB1 Q9Y478 10/20 0.66
ACVR1 Q04771 8/20 0.66
TGFBR1 P36897 5/20 0.66
ACVR1B P36896 5/20 0.66
BMPR1B O00238 5/20 0.66
ACVRL1 P37023 5/20 0.66
BMPR1A P36894 4/20 0.66
TGFBR2 P37173 3/20 0.66
BMPR2 Q13873 3/20 0.66
PRKAB2 O43741 6/20 0.53
PRKAG1 P54619 6/20 0.53
PRKAA2 P54646 6/20 0.53
PRKAA1 Q13131 6/20 0.53
PRKAG3 Q9UGI9 6/20 0.53
PRKAG2 Q9UGJ0 6/20 0.53
FLT1 P17948 6/20 0.53
FLT4 P35916 3/20 0.53
LCK P06239 4/20 0.50
SRC P12931 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30508268 0.83 KDR (0.55) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL5416682 0.82 KDR (0.67) KDRPRKAB1ACVR1TGFBR1PRKAB2
SCHEMBL3758736 0.79 MAP4K4 (0.57) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL31060220 0.79 PRKAB1 (1.00) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL6374645 0.78 KMO (0.61)
SCHEMBL13126019 0.77 KDR (0.76) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL29042049 0.76 FYN (0.65) ACVR1TGFBR1BMPR1BACVRL1BMPR1A
SCHEMBL26867136 0.75 ACVR1 (0.74) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL15996329 0.75 ACVR1 (1.00) KDRPRKAB1ACVR1TGFBR1ACVR1B
SCHEMBL17442229 0.74 ACVR1 (0.73) KDRPRKAB1ACVR1TGFBR1ACVR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed