SCHEMBL30508338

SCHEMBL30508338

COC(=O)c1cc(-c2ccc3nn(CCN4CCOCC4)cc3c2)cnc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
TBK1 Q9UHD2 6/20 0.50
IKBKE Q14164 5/20 0.50
BMPR1B O00238 5/20 0.46
BMPR1A P36894 5/20 0.46
TGFBR1 P36897 5/20 0.46
ACVRL1 P37023 5/20 0.46
ACVR1 Q04771 5/20 0.46
PIK3CA P42336 2/20 0.43
PIK3C3 Q8NEB9 1/20 0.42
AXL P30530 1/20 0.42
MERTK Q12866 1/20 0.42
SLC2A1 P11166 1/20 0.42
FGFR1 P11362 1/20 0.41
FGFR2 P21802 1/20 0.41
FGFR3 P22607 1/20 0.41
WNT1 P04628 1/20 0.40
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042097 1.00 HDAC3 (0.52) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL30508285 0.89 HDAC3 (0.55) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL30508316 0.89 HDAC3 (0.41) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL29041963 0.89 HDAC3 (0.41) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL30508377 0.83 BMPR1B (0.61) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL29041964 0.80 IRAK4 (0.48) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL30508232 0.80 IRAK4 (0.48) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL29152375 0.79 BMPR1B (0.64) TBK1IKBKEBMPR1BBMPR1ATGFBR1
SCHEMBL30508414 0.79 BMPR1B (0.64) TBK1IKBKEBMPR1BBMPR1ATGFBR1
SCHEMBL15681626 0.79 HDAC3 (0.57) HDAC3HDAC1HDAC2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
WO-2023198114-A1 ALK2 KINASE INHIBITOR 杭州邦顺制药有限公司 2023-10-19 WO disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed