SCHEMBL29041963

SCHEMBL29041963

COC(=O)c1cc(-c2ccc3nn(CCN4CCC(F)(F)CC4)cc3c2)cnc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.41
TBK1 Q9UHD2 5/20 0.39
IKBKE Q14164 4/20 0.39
CNR2 P34972 1/20 0.38
KIT P10721 1/20 0.38
MCHR1 Q99705 2/20 0.38
AXL P30530 1/20 0.37
MERTK Q12866 1/20 0.37
BMPR1B O00238 5/20 0.37
BMPR1A P36894 5/20 0.37
TGFBR1 P36897 5/20 0.37
ACVRL1 P37023 5/20 0.37
ACVR1 Q04771 5/20 0.37
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30508316 1.00 HDAC3 (0.41) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL30508200 0.90 HDAC3 (0.43) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL29042097 0.89 HDAC3 (0.52) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL30508338 0.89 HDAC3 (0.52) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL30508332 0.85 BMPR1B (0.51) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL30508285 0.78 HDAC3 (0.55) HDAC3HDAC1HDAC2PIK3C3TBK1
SCHEMBL29042061 0.77 BMPR1B (0.43) PIK3C3TBK1IKBKEAXLMERTK
SCHEMBL30508219 0.77 BMPR1B (0.43) PIK3C3TBK1IKBKEAXLMERTK
SCHEMBL30508377 0.76 BMPR1B (0.61) HDAC3HDAC1HDAC2TBK1IKBKE
SCHEMBL9960533 0.69 PIK3CA (0.48) TBK1IKBKEKITPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed