SCHEMBL30508285

SCHEMBL30508285

Nc1ncc(-c2ccc3nn(CCN4CCOCC4)cc3c2)cc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
IKBKE Q14164 4/20 0.51
TBK1 Q9UHD2 4/20 0.51
BMPR1B O00238 7/20 0.45
BMPR1A P36894 7/20 0.45
TGFBR1 P36897 7/20 0.45
ACVRL1 P37023 7/20 0.45
ACVR1 Q04771 7/20 0.45
PIK3CA P42336 1/20 0.43
PIK3C3 Q8NEB9 1/20 0.41
GRK5 P34947 1/20 0.40
ATR Q13535 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
MCHR1 Q99705 1/20 0.39
AXL P30530 1/20 0.39
MERTK Q12866 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042097 0.89 HDAC3 (0.52) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508338 0.89 HDAC3 (0.52) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508200 0.88 HDAC3 (0.43) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508377 0.84 BMPR1B (0.61) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508339 0.78 MET (0.44) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL29041963 0.78 HDAC3 (0.41) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508316 0.78 HDAC3 (0.41) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508336 0.77 ACVR1 (0.64) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL15681625 0.77 HDAC3 (0.61) HDAC3HDAC1HDAC2PIK3CAMCHR1
SCHEMBL30508238 0.76 LRRK2 (0.57) IKBKETBK1BMPR1BBMPR1ATGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
WO-2023198114-A1 ALK2 KINASE INHIBITOR 杭州邦顺制药有限公司 2023-10-19 WO disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed