SCHEMBL30512136

SCHEMBL30512136

O=C(O)c1cc(Nc2ncc3ccccc3n2)c[nH]1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 3/20 0.54
ROCK1 Q13464 1/20 0.45
BRAF P15056 3/20 0.40
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
DGAT1 O75907 1/20 0.39
MGAM O43451 1/20 0.38
CDK2 P24941 3/20 0.38
AURKA O14965 3/20 0.38
GSK3B P49841 2/20 0.38
MAPK1 P28482 1/20 0.38
GSK3A P49840 1/20 0.38
FDPS P14324 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK8 P45983 2/20 0.37
CDC7 O00311 1/20 0.37
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25881961 1.00 MAP3K5 (0.54) MAP3K5ROCK1BRAFCSNK2A2CSNK2B
SCHEMBL25881960 0.86 MAP3K5 (0.54) MAP3K5ROCK1BRAF
SCHEMBL30512112 0.86 MAP3K5 (0.54) MAP3K5ROCK1BRAFCDK2AURKA
SCHEMBL25879550 0.86 MAP3K5 (0.54) MAP3K5ROCK1BRAFCDK2AURKA
SCHEMBL30512103 0.83 MAP3K5 (0.50) MAP3K5ROCK1BRAFCDK2AURKA
SCHEMBL25881661 0.81 MAP3K5 (0.48) MAP3K5ROCK1BRAFCDK2FDPS
SCHEMBL25879895 0.80 BRAF (0.51) MAP3K5BRAFCDK2AURKAMAPK1
SCHEMBL25879889 0.80 HRH4 (0.50) MAP3K5CDK2
SCHEMBL30512108 0.80 BRAF (0.51) MAP3K5BRAFCDK2AURKAMAPK1
SCHEMBL25880449 0.78 HRH4 (0.53) MAP3K5CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed