SCHEMBL25880449

SCHEMBL25880449

CN1CC2CN(C(=O)c3cc(Nc4ncc5ccccc5n4)c[nH]3)CC2C1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 7/20 0.53
MAP3K5 Q99683 1/20 0.45
AXL P30530 2/20 0.43
CCNA2 P20248 6/20 0.42
CDK2 P24941 6/20 0.42
CDK7 P50613 6/20 0.42
CCNH P51946 6/20 0.42
MNAT1 P51948 6/20 0.42
CCNK O75909 5/20 0.42
CDK12 Q9NYV4 5/20 0.42
HCRTR2 O43614 2/20 0.41
HRH3 Q9Y5N1 2/20 0.39
VNN1 O95497 2/20 0.39
HCRTR1 O43613 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25879889 0.87 HRH4 (0.50) HRH4MAP3K5CDK2HRH3
SCHEMBL25882002 0.78 EGFR (0.48) MAP3K5AXLCCNA2CDK2
SCHEMBL30512114 0.78 EGFR (0.48) MAP3K5AXLCCNA2CDK2
SCHEMBL25881961 0.78 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL30512136 0.78 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL30512112 0.77 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL25881960 0.77 MAP3K5 (0.54) MAP3K5
SCHEMBL25879550 0.77 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL25880004 0.76 SYK (0.45) MAP3K5
SCHEMBL30512121 0.75 BRAF (0.46) MAP3K5AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed