SCHEMBL25879889

SCHEMBL25879889

CN1CCN(C(=O)c2cc(Nc3ncc4ccccc4n3)c[nH]2)CC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.50
HRH3 Q9Y5N1 1/20 0.50
MAP3K5 Q99683 1/20 0.47
SYK P43405 9/20 0.46
NUAK1 O60285 1/20 0.44
MAP4K1 Q92918 1/20 0.44
CCNT1 O60563 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
CDK9 P50750 1/20 0.44
ABL1 P00519 1/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
SRC P12931 1/20 0.43
PDGFRA P16234 1/20 0.43
MAPK14 Q16539 1/20 0.43
WEE1 P30291 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25880449 0.87 HRH4 (0.53) HRH4HRH3MAP3K5CDK2
SCHEMBL25880000 0.83 BRAF (0.46) MAP3K5MAP4K1PDGFRBPDGFRA
SCHEMBL30512121 0.83 BRAF (0.46) MAP3K5MAP4K1PDGFRBPDGFRA
SCHEMBL25882002 0.82 EGFR (0.48) MAP3K5SYKMAP4K1CDK2WEE1
SCHEMBL30512114 0.82 EGFR (0.48) MAP3K5SYKMAP4K1CDK2WEE1
SCHEMBL25880004 0.80 SYK (0.45) MAP3K5SYKMAP4K1
SCHEMBL30512136 0.80 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL25881961 0.80 MAP3K5 (0.54) MAP3K5CDK2
SCHEMBL30512112 0.79 MAP3K5 (0.54) MAP3K5SYKCDK2
SCHEMBL25879550 0.79 MAP3K5 (0.54) MAP3K5SYKCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed