SCHEMBL30516118

SCHEMBL30516118

O=C(NO)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.56
HDAC1 Q13547 8/20 0.56
HDAC3 O15379 6/20 0.49
HDAC2 Q92769 5/20 0.49
SLC6A3 Q01959 1/20 0.48
KCNH2 Q12809 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48
HDAC4 P56524 1/20 0.47
HDAC8 Q9BY41 1/20 0.46
TRPV1 Q8NER1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045114 1.00 HDAC6 (0.56) HDAC6HDAC1HDAC3HDAC2SLC6A3
SCHEMBL2224785 0.84 P2RX7 (0.49) SLC6A3KCNH2TAAR1TRPV1
SCHEMBL3550941 0.84 BAZ2B (0.51) HDAC6HDAC2SLC6A3KCNH2TAAR1
Hydrochloric Acid SCHEMBL28637532 0.83 P2RX7 (0.47) SLC6A3KCNH2TAAR1TRPV1
SCHEMBL29827745 0.82 P4HTM (0.60) KCNH2TRPV1
SCHEMBL22387735 0.82 HDAC6 (0.61) HDAC6HDAC1HDAC3HDAC2HDAC8
SCHEMBL13701813 0.81 LMNA (0.46) SLC6A3KCNH2TAAR1TRPV1
SCHEMBL6140597 0.81 TRPV4 (0.52) SLC6A3KCNH2TAAR1HDAC4TRPV1
SCHEMBL3544820 0.80 PTPN1 (0.47) SLC6A3KCNH2TAAR1TRPV1
SCHEMBL22915155 0.80 HSP90AA1 (0.49) HDAC6HDAC4TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN disclosed