SCHEMBL30516492

SCHEMBL30516492

O=C1CN(C(=O)CCBr)c2ccccc2N1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.70
CASP2 P42575 1/20 0.70
KMT2A Q03164 2/20 0.63
ALDH1A1 P00352 4/20 0.60
GAA P10253 2/20 0.60
LMNA P02545 1/20 0.60
KDM4E B2RXH2 1/20 0.60
HTT P42858 2/20 0.59
USP2 O75604 1/20 0.58
MAPT P10636 1/20 0.58
HPGD P15428 1/20 0.58
PKM P14618 1/20 0.57
MEN1 O00255 1/20 0.57
MAPK1 P28482 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
TSHR P16473 1/20 0.56
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
SHMT2 P34897 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29064837 1.00 CASP3 (0.70) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL24335274 0.87 CASP3 (0.72) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL30516491 0.87 CASP3 (0.72) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL24335146 0.87 CASP3 (0.72) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL24335266 0.84 CASP3 (0.68) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL30516505 0.84 CASP3 (0.68) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL25430532 0.84 CASP3 (0.76) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL29580313 0.83 CASP3 (0.67) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL11035331 0.82 CASP3 (1.00) CASP3CASP2KMT2AALDH1A1GAA
SCHEMBL24335192 0.82 KMT2A (0.66) CASP3CASP2KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116528867-A Compounds for the treatment of Alzheimer's disease 艾伯塔大学理事会 2023-08-01 CN disclosed