SCHEMBL30516518

SCHEMBL30516518

CC(O)(c1nccs1)C(O)Cc1cccc(Oc2ncnc3[nH]ccc23)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.45
TNNI3K Q59H18 2/20 0.45
MAP3K14 Q99558 10/20 0.44
KDR P35968 2/20 0.40
BRAF P15056 1/20 0.40
MAPK14 Q16539 1/20 0.40
CIT O14578 1/20 0.37
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28657455 1.00 TRPA1 (0.45) TRPA1TNNI3KMAP3K14KDRBRAF
SCHEMBL28639382 0.78 MAP3K14 (0.68) MAP3K14
SCHEMBL30516482 0.78 MAP3K14 (0.68) MAP3K14
SCHEMBL4548935 0.64 KDR (0.69) TRPA1TNNI3KKDRBRAFMAPK14
SCHEMBL23072725 0.60 TRPA1 (0.55) TRPA1TNNI3KKDRBRAFMAPK14
SCHEMBL20439521 0.60 TRPA1 (0.55) TRPA1TNNI3KKDRBRAFMAPK14
SCHEMBL28524919 0.60 CTSA (0.40)
SCHEMBL20437215 0.60 ITGB3 (0.53) TRPA1TNNI3KKDRBRAFMAPK14
SCHEMBL4548932 0.60 KDR (0.70) TRPA1TNNI3KKDRBRAFMAPK14
SCHEMBL2882091 0.59 TRPA1 (0.75) TRPA1TNNI3KKDRBRAFMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112794855-B Preparation method and application of N-aryl pyrimidine-4-amine derivative 中国药科大学 2023-07-28 CN disclosed