SCHEMBL28524919

SCHEMBL28524919

CC(C)(C)NC(=O)Oc1cccc(C[C@@H](O)c2nccs2)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSA P10619 7/20 0.40
ALOX5 P09917 1/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ACHE P22303 2/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BCHE P06276 1/20 0.36
PTPRB P23467 1/20 0.36
FFAR1 O14842 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28531299 0.89 CTSA (0.39) CTSAALOX5NPC1RAB9AACHE
SCHEMBL28530968 0.82 MEN1 (0.46) CTSAALOX5NPC1RAB9AFFAR1
SCHEMBL28530965 0.82 MEN1 (0.46) CTSAALOX5NPC1RAB9AFFAR1
SCHEMBL28524920 0.77 AURKA (0.44)
SCHEMBL29643010 0.77 AURKA (0.44)
SCHEMBL28101915 0.75 ACHE (0.41) ACHEBCHE
SCHEMBL28524607 0.75 ACHE (0.41) ACHEBCHE
SCHEMBL27765570 0.74 TSHR (0.43) ACHESMN1; SMN2BCHE
SCHEMBL20541076 0.73 ACHE (0.43) ACHEBCHE
SCHEMBL27605135 0.73 LOXL2 (0.48) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112437675-A Antibody drug conjugates for ablating hematopoietic stem cells 诺华股份有限公司 2021-03-02 CN disclosed