SCHEMBL30516692

SCHEMBL30516692

COC(=O)c1cc(-c2ccc(F)cn2)cc(OCC(F)F)c1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
LMNA P02545 1/20 0.37
GABRA5 P31644 1/20 0.37
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
TGFBR1 P36897 3/20 0.35
TGFBR2 P37173 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
P2RX7 Q99572 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24478734 1.00 NPC1 (0.38) NPC1CASP3RAB9ASMN1; SMN2SENP8
SCHEMBL24478751 0.88 LDHA (0.42) NPC1GABRA5P2RX7NR1I2LDHA
SCHEMBL30516696 0.88 LDHA (0.42) NPC1GABRA5P2RX7NR1I2LDHA
SCHEMBL30516698 0.74 KDM4E (0.41) ALDH1A1HPGDTSHRCASP1HSD17B10
SCHEMBL24478766 0.74 KDM4E (0.41) ALDH1A1HPGDTSHRCASP1HSD17B10
SCHEMBL16598552 0.74 ALDH1A1 (0.45) LMNASLC6A4SLC6A3ALDH1A1TSHR
SCHEMBL24525359 0.73 NPC1 (0.51) NPC1CASP3RAB9ASMN1; SMN2SENP8
SCHEMBL29654515 0.73 NPC1 (0.51) NPC1CASP3RAB9ASMN1; SMN2SENP8
SCHEMBL23460499 0.73 TDP1 (0.50) NPC1CASP3RAB9ASMN1; SMN2SENP8
SCHEMBL25486957 0.70 NPC1 (0.41) NPC1CASP3RAB9ASMN1; SMN2SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601149-A Aminoquinazoline derivatives as P2X3 inhibitors 奇斯药制品公司 2023-08-15 CN disclosed