SCHEMBL30519087

SCHEMBL30519087

CCCCCCC#Cc1cncc(-c2nnc(S)n2C)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.39
CHRNA3 P32297 6/20 0.39
MAPT P10636 2/20 0.38
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
GRM5 P41594 1/20 0.35
CHRNA2 Q15822 3/20 0.32
CHRNA4 P43681 2/20 0.32
CHRNB4 P30926 1/20 0.32
FFAR1 O14842 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25333101 1.00 CHRNB2 (0.39) CHRNB2CHRNA3MAPTSAE1UBA2
SCHEMBL25932870 0.85 CHRNB2 (0.38) CHRNB2CHRNA3MAPTSAE1UBA2
SCHEMBL13856833 0.78 NPC1 (0.48) MAPT
SCHEMBL13856839 0.77 KMT2A (0.42) MAPTGRM5
SCHEMBL25334094 0.72 RAB9A (0.40) MAPTSAE1UBA2GRM5
SCHEMBL2860394 0.70 HPGD (0.44) CHRNB2CHRNA3HSD11B1
SCHEMBL15544407 0.68 KCNH2 (0.45) CHRNB2MAPTSAE1UBA2GRM5
SCHEMBL7453866 0.67 CYP2A6 (0.41)
SCHEMBL17079717 0.66 MAPT (0.58) MAPTSAE1UBA2FFAR1FFAR4
SCHEMBL1934205 0.66 KCNH2 (0.42) CHRNB2CHRNA3MAPTSAE1UBA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4472630-A2 SELECTIVE AGENTS TARGETING MYCOBACTERIUM TUBERCULOSIS University of Mississippi (US) 2024-12-11 EP disclosed
WO-2023147571-A2 SELECTIVE AGENTS TARGETING MYCOBACTERIUM TUBERCULOSIS UNIVERSITY OF MISSISSIPPI (US) 2023-08-03 WO disclosed