SCHEMBL30529792

SCHEMBL30529792

Cc1ncc2c(n1)NC(=O)N(C1CCOCC1)C2

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
JAK2 O60674 5/20 0.39
PRKDC P78527 2/20 0.36
PIK3CG P48736 1/20 0.36
PRKCB P05771 1/20 0.34
PDE9A O76083 4/20 0.33
GABRA1 P14867 1/20 0.33
PDE1C Q14123 2/20 0.33
PIK3CD O00329 1/20 0.33
JAK1 P23458 1/20 0.33
PDE1B Q01064 1/20 0.33
MAPK1 P28482 2/20 0.33
HCAR1 Q9BXC0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30853317 0.76 FGFR4 (0.44) PIK3CAMTORJAK2PRKDCPIK3CG
SCHEMBL25462291 0.73 HPGD (0.41) MAPK1
SCHEMBL28655766 0.68 PIK3CA (0.35) PIK3CAMTORPIK3CGPIK3CD
SCHEMBL26160595 0.65 JAK2 (0.57) MTORJAK2PRKDCJAK1HCAR1
SCHEMBL4044760 0.65 PDE3B (0.48) PIK3CG
SCHEMBL152295 0.64 MTOR (0.59) PIK3CAMTORJAK2PRKDC
SCHEMBL29522157 0.64 MTOR (0.59) PIK3CAMTORJAK2PRKDC
SCHEMBL14042006 0.64 PDE3B (0.46)
SCHEMBL151621 0.64 MTOR (0.57) PIK3CAMTORJAK2PRKDC
SCHEMBL30030188 0.63 MAPK8 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113912608-B Pyrimidopyrimidinone derivatives, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2023-07-14 CN disclosed