SCHEMBL30543333

SCHEMBL30543333

O=C1NCc2c1cccc2-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.52
KDR P35968 10/20 0.49
ROCK2 O75116 5/20 0.46
PIM1 P11309 5/20 0.45
ROCK1 Q13464 5/20 0.45
CLK4 Q9HAZ1 5/20 0.45
DYRK1A Q13627 4/20 0.45
CDK5 Q00535 2/20 0.45
CSNK1A1 P48729 1/20 0.45
LRRK2 Q5S007 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
PIK3CD O00329 1/20 0.45
PIK3CA P42336 1/20 0.45
PIK3CB P42338 1/20 0.45
MAP4K4 O95819 4/20 0.45
AURKB Q96GD4 4/20 0.45
RET P07949 3/20 0.45
RPS6KB1 P23443 3/20 0.45
PLK4 O00444 3/20 0.45
FLT4 P35916 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30775205 0.85 KDR (0.49) KDRROCK2PIM1ROCK1CLK4
SCHEMBL30775209 0.82 CNR2 (0.58) CNR2KDR
SCHEMBL30775367 0.81 L3MBTL1 (0.52) PIM1ROCK1CLK4DYRK1ACDK5
SCHEMBL30543359 0.81 KDR (0.50) KDRROCK2PIM1ROCK1MAP4K4
SCHEMBL30331758 0.75 PARP10 (0.69) KDRROCK2PIM1ROCK1CLK4
SCHEMBL19608227 0.74 PIK3CD (0.64) KDRROCK2PIM1ROCK1CLK4
SCHEMBL1333209 0.74 KDR (0.57) KDRROCK2PIM1ROCK1CLK4
SCHEMBL28223904 0.74 PIK3CD (0.64) KDRROCK2PIM1ROCK1CLK4
SCHEMBL30598685 0.72 TBK1 (0.56) PIK3CDPIK3CAPIK3CBMKNK2TBK1
SCHEMBL28241795 0.72 OGA (0.50) KDRCLK4DYRK1BPIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116496246-A Isoindoline compound, preparation method, pharmaceutical composition and application 中国药科大学 2023-07-28 CN claimed
CN-116496246-A Isoindoline compound, preparation method, pharmaceutical composition and application 中国药科大学 2023-07-28 CN disclosed