SCHEMBL30547733

SCHEMBL30547733

CC(C)c1ccc2c(c1)cc(C(N)=O)n2C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
MCL1 Q07820 2/20 0.45
PHGDH O43175 6/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC9A1 P19634 1/20 0.42
CLK1 P49759 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
THRB P10828 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
JAK3 P52333 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
AHR P35869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12894673 1.00 KDM4E (0.45) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL13895694 0.88 SLC9A1 (0.42) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL9613270 0.86 HSD17B10 (0.62) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL30790917 0.86 HSD17B10 (0.62) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL13881405 0.86 KDM4E (0.46) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL9613264 0.79 THRB (0.61) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL28238032 0.79 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL6086802 0.79 CLK1 (0.61) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL13415456 0.78 RXFP1 (0.62) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL4744999 0.78 KDM4E (0.73) KDM4EALDH1A1HPGDHSD17B10MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423435-B1 SUBSTITUTED INDOLE MCL-1 INHIBITORS UNIV VANDERBILT (US) 2023-08-23 EP disclosed