SCHEMBL30587462

SCHEMBL30587462

COC(=O)c1ncn(Cc2ncccc2F)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 2/20 0.41
HDAC1 Q13547 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
NOTUM Q6P988 1/20 0.38
RIPK1 Q13546 7/20 0.38
ADORA2A P29274 1/20 0.38
HDAC4 P56524 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
EED O75530 1/20 0.36
SUZ12 Q15022 1/20 0.36
EZH2 Q15910 1/20 0.36
KLKB1 P03952 1/20 0.36
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18367255 1.00 SLC40A1 (0.41) SLC40A1HDAC1HDAC6NOTUMRIPK1
SCHEMBL18367236 0.86 ADORA2A (0.40) NOTUMRIPK1ADORA2AKLKB1KDM4E
SCHEMBL18367259 0.85 NOTUM (0.46) SLC40A1NOTUMRIPK1KLKB1KDM4E
SCHEMBL30587508 0.85 NOTUM (0.46) SLC40A1NOTUMRIPK1KLKB1KDM4E
SCHEMBL18367248 0.84 SLC40A1 (0.42) SLC40A1HDAC1HDAC6RIPK1HDAC4
SCHEMBL22736832 0.83 CA5A (0.42) HDAC1HDAC6NOTUMRIPK1EED
SCHEMBL18366884 0.82 RIPK1 (0.52) HDAC1HDAC6RIPK1HDAC4HDAC2
SCHEMBL30587636 0.82 RIPK1 (0.52) HDAC1HDAC6RIPK1HDAC4HDAC2
SCHEMBL18366888 0.80 RIPK1 (0.46) HDAC1HDAC6NOTUMRIPK1HDAC4
SCHEMBL30092641 0.80 RIPK1 (0.46) HDAC1HDAC6NOTUMRIPK1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111269221-B Bicyclic lactams and methods of use thereof 豪夫迈·罗氏有限公司 2023-09-26 CN disclosed