SCHEMBL30593191

SCHEMBL30593191

CCOC(=O)c1c(OCc2ccc(OC)cc2)cc(Cl)nc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
POLB P06746 1/20 0.53
MAOB P27338 2/20 0.52
KMT2A Q03164 3/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAPT P10636 3/20 0.46
PTPN11 Q06124 1/20 0.45
PDE4D Q08499 1/20 0.45
ALDH1A1 P00352 4/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
USP2 O75604 1/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25151518 1.00 GAA (0.53) GAAPOLBMAOBKMT2ACASP3
SCHEMBL26608385 0.87 MTNR1A (0.46) GAAPOLBMAOBKMT2ACASP3
SCHEMBL26601614 0.87 POLB (0.49) GAAPOLBMAOBKMT2ACASP3
SCHEMBL26601686 0.87 RAB9A (0.50) GAAKMT2AMAPTALDH1A1HPGD
SCHEMBL31336208 0.87 RAB9A (0.50) GAAKMT2AMAPTALDH1A1HPGD
SCHEMBL26601891 0.86 NPSR1 (0.43) GAAPOLBMAOBKMT2ACASP3
SCHEMBL24772939 0.81 GAA (0.53) GAAPOLBMAPTALDH1A1HPGD
SCHEMBL14966627 0.80 MAOB (0.48) GAAPOLBMAOBMAPTPTPN11
SCHEMBL30887705 0.79 GAA (0.52) GAAPOLBKMT2ACASP3SENP8
SCHEMBL31747868 0.78 GAA (0.44) GAAPOLBMAOBKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4511115-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN Vertex Pharmaceuticals Incorporated (US) 2025-02-26 EP disclosed
WO-2023205468-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-26 WO disclosed