SCHEMBL30593308

SCHEMBL30593308

NC(=O)N1CCc2ccc(-c3ccccc3)cc2C1c1c[nH]c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.46
CCR2 P41597 2/20 0.42
KDM4E B2RXH2 2/20 0.40
BRD4 O60885 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
CREBBP Q92793 1/20 0.40
HSD11B1 P28845 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
PDE4D Q08499 2/20 0.39
ECE1 P42892 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
KCNA3 P22001 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30593227 0.92 ECE1 (0.44) KIF11CCR2KDM4EBRD4ALDH1A1
SCHEMBL30593296 0.88 DRD2 (0.41) KIF11KDM4EHSD11B1LMNAMAPT
SCHEMBL29084839 0.88 DRD2 (0.41) KIF11KDM4EHSD11B1LMNAMAPT
SCHEMBL30593300 0.86 DRD2 (0.49) KIF11KDM4EBRD4ALDH1A1POLB
SCHEMBL31083691 0.84 KIF11 (0.41) KIF11CCR2KDM4EBRD4ALDH1A1
SCHEMBL31070623 0.83 ECE1 (0.40) KIF11CCR2KDM4EBRD4ALDH1A1
SCHEMBL31083744 0.82 PDE4D (0.45) KIF11HSD11B1LMNAMAPTPDE4D
SCHEMBL31083723 0.82 KIF11 (0.41) KIF11CCR2KDM4EBRD4ALDH1A1
SCHEMBL31083762 0.82 KIF11 (0.41) KIF11CCR2KDM4EBRD4ALDH1A1
SCHEMBL31083773 0.82 PDE4D (0.47) KIF11HSD11B1LMNAMAPTPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed