SCHEMBL30593296

SCHEMBL30593296

NC(=O)N1CCc2ccccc2C1c1c[nH]c2ccc(-c3ccccc3)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41
NR4A2 P43354 1/20 0.41
KIF11 P52732 7/20 0.39
HTR6 P50406 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
ICMT O60725 1/20 0.39
CNR2 P34972 1/20 0.38
HSD11B1 P28845 1/20 0.38
IKBKB O14920 1/20 0.37
NOS1 P29475 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29084839 1.00 DRD2 (0.41) DRD2DRD1DRD5NR4A2KIF11
SCHEMBL31070497 0.89 NR4A2 (0.42) NR4A2HTR6ICMTCNR2IKBKB
SCHEMBL30593227 0.88 ECE1 (0.44) DRD2DRD1DRD5KIF11HSD11B1
SCHEMBL30593308 0.88 KIF11 (0.46) KIF11HSD11B1KDM4ELMNAMAPT
SCHEMBL31083752 0.87 KIF11 (0.49) NR4A2KIF11HTR6ICMTHSD11B1
SCHEMBL30593317 0.87 HSD11B1 (0.43) ICMTHSD11B1
SCHEMBL31083748 0.87 KIF11 (0.48) KIF11HSD11B1MAPT
SCHEMBL31083802 0.87 ECE1 (0.38) KIF11HTR6HSD11B1
SCHEMBL31083737 0.86 GRM4 (0.41) DRD2DRD1DRD5KIF11HSD11B1
SCHEMBL30593291 0.86 KIF11 (0.52) DRD2DRD1DRD5KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed