Bicarbonate

Bicarbonate

SCHEMBL3059503

CCCC(=O)OC(C)c1cc([N+](=O)[O-])ccc1O.O=C(O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL9 O00512 1/20 0.48
CTNNB1 P35222 1/20 0.48
GAA P10253 4/20 0.47
MAPT P10636 4/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
GRM8 O00222 1/20 0.42
GRM4 Q14833 1/20 0.42
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
KDM4E B2RXH2 2/20 0.41
GLA P06280 1/20 0.41
TDP1 Q9NUW8 2/20 0.40
COMT P21964 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26740 0.83 BCL9 (0.49) BCL9CTNNB1GAAMAPTL3MBTL1
SCHEMBL26741 0.83 BCL9 (0.49) BCL9CTNNB1GAAMAPTL3MBTL1
SCHEMBL26739 0.82 BCL9 (0.50) BCL9CTNNB1MAPTPOLBSMN1; SMN2
SCHEMBL10061896 0.80 MAPT (0.47) GAAMAPTL3MBTL1POLBSMN1; SMN2
SCHEMBL4380543 0.77 BCL9 (0.62) BCL9CTNNB1GAAMAPTL3MBTL1
SCHEMBL29402294 0.77 BCL9 (0.62) BCL9CTNNB1GAAMAPTL3MBTL1
SCHEMBL8041378 0.74 SMN1; SMN2 (0.51) GAAMAPTL3MBTL1POLBSMN1; SMN2
SCHEMBL25823 0.73 CYSLTR2 (0.41) BCL9CTNNB1MAPTPOLBSMN1; SMN2
SCHEMBL25822 0.73 CYSLTR2 (0.41) BCL9CTNNB1MAPTPOLBSMN1; SMN2
SCHEMBL4369630 0.72 GAA (0.50) GAAMAPTL3MBTL1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790708-B2 Prodrugs of GABA analogs, compositions and uses thereof XENOPORT, INC. (US) 2010-09-07 US disclosed
US-20070010453-A1 Prodrugs of GABA analogs, compositions and uses thereof XENOPORT, INC. 2007-01-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070010453-A1 Prodrugs of GABA analogs, compositions and uses thereof GABRB1, GABRB2, GABRB3 BCL9 2365/4885CTNNB1 4448/4885GAA 439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.