E-Flupentixol

E-Flupentixol

SCHEMBL30596168

OCCN1CCN(CCC=C2c3ccccc3Sc3ccc(C(F)(F)F)cc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 1.00
USP2 O75604 6/20 1.00
SIGMAR1 Q99720 5/20 1.00
CYP2D6 P10635 5/20 1.00
MAPK1 P28482 5/20 1.00
TP53 P04637 5/20 1.00
CYP1A2 P05177 4/20 1.00
NFKB1 P19838 4/20 1.00
CYP2C19 P33261 3/20 1.00
THPO P40225 3/20 1.00
TSHR P16473 3/20 1.00
KCNK2 O95069 2/20 1.00
LMNA P02545 8/20 0.98
MEN1 O00255 7/20 0.98
KMT2A Q03164 7/20 0.98
RAD52 P43351 3/20 0.98
GMNN O75496 3/20 0.98
PMP22 Q01453 3/20 0.98
TDP1 Q9NUW8 3/20 0.98
HTR1A P08908 4/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Z-Flupentixol SCHEMBL34200 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
E-Flupentixol SCHEMBL145726 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
E-Flupentixol SCHEMBL29598791 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
Z-Flupentixol SCHEMBL29361845 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
E-Flupentixol SCHEMBL414352 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
Z-Flupentixol SCHEMBL29620416 1.00 CYP3A4 (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
E-Flupentixol SCHEMBL11427109 0.99 LMNA (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
Z-Flupentixol SCHEMBL719323 0.99 LMNA (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
E-Flupentixol SCHEMBL1230220 0.99 LMNA (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1
Z-Flupentixol SCHEMBL1153162 0.99 LMNA (1.00) CYP3A4USP2SIGMAR1CYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116804000-A Specific palmitoyl transferase inhibitor and application thereof 苏州大学 2023-09-26 CN claimed
CN-116804000-A Specific palmitoyl transferase inhibitor and application thereof 苏州大学 2023-09-26 CN disclosed