SCHEMBL30608922

SCHEMBL30608922

FCCCN1CC[C@H](Nc2cnccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.41
HRH2 P25021 2/20 0.41
ROCK2 O75116 8/20 0.37
CCR2 P41597 4/20 0.37
ROCK1 Q13464 4/20 0.37
AXL P30530 1/20 0.36
FLT3 P36888 1/20 0.36
TYRO3 Q06418 1/20 0.36
MERTK Q12866 1/20 0.36
ESR1 P03372 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP2D6 P10635 1/20 0.35
CHEK1 O14757 1/20 0.35
CHEK2 O96017 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30608962 0.89 ESR1 (0.38) HRH1HRH2ESR1KCNH2CYP2D6
SCHEMBL30608923 0.84 ROCK2 (0.46) HRH1HRH2ROCK2CCR2ROCK1
SCHEMBL30608972 0.82 NOS2 (0.47) HRH1HRH2DRD2DRD3
SCHEMBL25851871 0.81 ESR1 (0.36) HRH1HRH2AXLFLT3TYRO3
SCHEMBL25851884 0.81 ESR1 (0.36) HRH1HRH2AXLFLT3TYRO3
SCHEMBL25494073 0.79 HRH2 (0.42) HRH1HRH2ROCK2CCR2ROCK1
SCHEMBL30346597 0.79 HRH2 (0.42) HRH1HRH2ROCK2CCR2ROCK1
SCHEMBL23098104 0.78 HRH4 (0.47) AXLCHEK1CHEK2
SCHEMBL30422610 0.72 ROCK2 (0.43) ROCK2CCR2ROCK1
SCHEMBL30346693 0.70 KDM4E (0.44) ESR1KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116964049-A Estrogen receptor modulators 里科瑞尔姆IP控股有限责任公司 2023-10-27 CN disclosed