SCHEMBL30627140

SCHEMBL30627140

FC(F)(F)c1cccc(-c2cccnc2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.57
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
PTK2 Q05397 1/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP19A1 P11511 2/20 0.46
PTGS2 P35354 2/20 0.45
NOTUM Q6P988 1/20 0.44
DYRK1A Q13627 1/20 0.44
TGFBR1 P36897 1/20 0.44
AXL P30530 2/20 0.44
MKNK1 Q9BUB5 2/20 0.44
MKNK2 Q9HBH9 2/20 0.44
PBRM1 Q86U86 1/20 0.44
MEN1 O00255 1/20 0.43
PSIP1 O75475 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRG2 P18507 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9007781 0.83 CYP2A6 (0.62) CYP2A6HSP90AA1HSP90AB1PTK2ALDH1A1
SCHEMBL2732457 0.83 CYP2A6 (0.62) CYP2A6HSP90AA1HSP90AB1PTK2ALDH1A1
SCHEMBL30419470 0.83 CYP2A6 (0.47) CYP2A6HSP90AA1HSP90AB1PTK2ALDH1A1
SCHEMBL19384206 0.82 NOTUM (0.46) NOTUMTGFBR1GABRA1GABRG2GABRB3
SCHEMBL3194702 0.81 CYP2A6 (0.74) CYP2A6HSP90AA1HSP90AB1PTK2ALDH1A1
SCHEMBL12278984 0.80 HPGDS (0.50) CYP2A6ALDH1A1CYP3A4CYP19A1TGFBR1
SCHEMBL3381636 0.80 MEN1 (0.60) NOTUMMEN1GABRA1GABRG2GABRB3
SCHEMBL12278291 0.78 MEN1 (0.47) CYP2A6ALDH1A1CYP1A2CYP3A4CYP19A1
SCHEMBL2183687 0.77 IDH1 (0.41) CYP2A6PTGS2TGFBR1MKNK1MEN1
SCHEMBL19384193 0.77 CYP11B2 (0.42) NOTUMTGFBR1GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116867758-A IRAK degradation agents and uses thereof 凯麦拉医疗公司 2023-10-10 CN disclosed