SCHEMBL30628

SCHEMBL30628

COc1cccc(C(=O)c2ccc(C3=CCCC(CNS(C)(=O)=O)=C3)s2)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 10/20 0.43
HSD17B1 P14061 9/20 0.43
ALDH1A1 P00352 2/20 0.38
STS P08842 2/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
USP2 O75604 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31148 0.88 HSD17B1 (0.47) HSD17B2HSD17B1
SCHEMBL29570 0.70 HSD17B1 (0.71) HSD17B2HSD17B1
SCHEMBL18195278 0.69 HSD17B2 (0.65) HSD17B2HSD17B1MAPK13MAPK12MAPK11
SCHEMBL23779 0.69 HSD17B2 (0.67) HSD17B2HSD17B1HDAC6
SCHEMBL23125 0.69 HSD17B2 (0.65) HSD17B2HSD17B1ALDH1A1NPC1HPGD
SCHEMBL31108 0.67 HSD17B1 (0.50) HSD17B2HSD17B1
SCHEMBL24822 0.66 HDAC6 (0.56) HSD17B2HSD17B1MAPK13MAPK12MAPK11
SCHEMBL10395539 0.65 CES2 (0.59) ALDH1A1STSNPC1HPGDRAB9A
SCHEMBL30620 0.65 HSD17B2 (0.58) HSD17B2HSD17B1HDAC6
SCHEMBL23339 0.65 HSD17B2 (0.66) HSD17B2HSD17B1MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed