SCHEMBL30632573

SCHEMBL30632573

CCn1c(N)c(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c(=O)n(CC)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.52
KMT2A Q03164 7/20 0.52
RAB9A P51151 3/20 0.52
NPC1 O15118 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
STAT1 P42224 1/20 0.52
KDM4E B2RXH2 4/20 0.52
HPGD P15428 4/20 0.51
ALDH1A1 P00352 3/20 0.51
NFE2L2 Q16236 1/20 0.50
CYP1A2 P05177 2/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
MAPT P10636 5/20 0.48
TP53 P04637 4/20 0.48
GAA P10253 3/20 0.48
CYP2C9 P11712 2/20 0.48
PDE4D Q08499 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28460284 0.92 FDPS (0.50) MEN1KMT2AHPGDALDH1A1
SCHEMBL28452461 0.92 MEN1 (0.46) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL7730987 0.90 ADORA2A (0.51) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL7730989 0.90 ADORA2A (0.51) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL28458573 0.88 FDPS (0.44) MEN1KMT2AKDM4EHPGDALDH1A1
SCHEMBL28377498 0.87 ALDH1A1 (0.44) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL28371613 0.87 ALDH1A1 (0.44) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL28429042 0.86 HDAC3 (0.39) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL28372708 0.86 PDE4D (0.45) MEN1KMT2ASMN1; SMN2KDM4EHPGD
SCHEMBL28887208 0.83 ALDH1A1 (0.42) MEN1KMT2ARAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088882-A Method for preparing high-purity itraconazole intermediate 山东新华制药股份有限公司 2023-11-21 CN claimed
CN-117088882-A Method for preparing high-purity itraconazole intermediate 山东新华制药股份有限公司 2023-11-21 CN disclosed
CN-117088882-A Method for preparing high-purity itraconazole intermediate 山东新华制药股份有限公司 2023-11-21 CN disclosed
CN-117024428-A Novel method for synthesizing itratheophylline 山东新华制药股份有限公司 2023-11-10 CN disclosed