SCHEMBL30690789

SCHEMBL30690789

Cc1ccc(NC(=O)OC(C)(C)C)cc1NC(=O)c1cnc2c(c1)cc(I)n2COCC[Si](C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.38
RORC P51449 4/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
KIT P10721 4/20 0.35
CSF1R P07333 1/20 0.35
HSF1 Q00613 3/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC6 Q9UBN7 2/20 0.34
PIR O00625 1/20 0.34
GSK3B P49841 1/20 0.34
EGFR P00533 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC10 Q969S8 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30690835 0.92 HDAC1 (0.36) RORCHDAC1HDAC6EGFRHDAC3
SCHEMBL30690786 0.81 FGFR1 (0.38) BRAFRORCKITHDAC1HDAC3
SCHEMBL30690642 0.77 CSF1R (0.41) RORCKITCSF1RHDAC1GSK3B
SCHEMBL30690782 0.75 ABL1 (0.32) HDAC1HDAC3
SCHEMBL30690811 0.75 DYRK1A (0.38) RORCKITCSF1RHDAC1GSK3B
SCHEMBL30690630 0.74 NPC1 (0.39)
SCHEMBL30690639 0.74 GSK3B (0.38) RORCKITCSF1RHDAC1GSK3B
SCHEMBL30690647 0.73 DYRK1A (0.41) RORCKITCSF1RGSK3BNAMPT
SCHEMBL14026831 0.72 BRAF (0.52) BRAFKITCSF1REGFRNAMPT
SCHEMBL30690763 0.71 GSK3B (0.36) HDAC1GSK3BHDAC3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023247593-A1 PYRROLOPYRIDINE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2023-12-28 WO disclosed