SCHEMBL30711998

SCHEMBL30711998

Cn1ncc2cc(C#N)c(O)nc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.34
HTT P42858 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
GLA P06280 1/20 0.33
MAPK1 P28482 1/20 0.33
KDM1A O60341 1/20 0.32
CDK2 P24941 1/20 0.32
CACNA1H O95180 3/20 0.32
CYP11B2 P19099 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
TP53 P04637 2/20 0.32
CSNK2A1 P68400 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23357465 1.00 MAPT (0.36) MAPTPOLBHTTSMN1; SMN2CYP1A2
SCHEMBL27072904 0.79 KDM4E (0.45) KDM4EALDH1A1IRAK4GAA
SCHEMBL30711996 0.79 ALDH1A1 (0.41) MAPTPOLBSMN1; SMN2CYP1A2CYP2C19
SCHEMBL23357368 0.79 ALDH1A1 (0.41) MAPTPOLBSMN1; SMN2CYP1A2CYP2C19
SCHEMBL5961491 0.73 ADORA2A (0.38) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL25386715 0.73 MEN1 (0.33) MAPTHTTSMN1; SMN2KDM4EALDH1A1
SCHEMBL20674173 0.71 HPGD (0.41) POLBHTTKDM4EALDH1A1HPGD
SCHEMBL16887703 0.70 TP53 (0.43) CYP11B2IRAK4TP53
SCHEMBL22337069 0.70 CYP11B2 (0.33) MAPTKDM1ACYP11B2TP53
SCHEMBL25881445 0.70 S1PR2 (0.36) MAPTALDH1A1MAPK1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110869363-B 5-membered and bicyclic heterocyclic amides as ROCK inhibitors 百时美施贵宝公司 2024-01-05 CN disclosed