SCHEMBL30714719

SCHEMBL30714719

Cc1ncc(COc2ccc3nn(C)c(C(=O)NC(C)(CO)C(N)=O)c3c2)o1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.33
RAB9A P51151 6/20 0.33
MAPT P10636 2/20 0.33
MCHR1 Q99705 7/20 0.33
POLB P06746 1/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSP90AA1 P07900 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30714623 0.90 MCHR1 (0.34) NPC1RAB9AMAPTMCHR1POLB
SCHEMBL26874836 0.85 MCHR1 (0.37) NPC1RAB9AMAPTMCHR1POLB
SCHEMBL30714551 0.84 ALOX5AP (0.39)
SCHEMBL30714568 0.84 MCHR1 (0.35) MCHR1SMN1; SMN2
SCHEMBL30714580 0.83 CYP11B2 (0.37) MCHR1SMN1; SMN2
SCHEMBL30714654 0.83 MCHR1 (0.34) NPC1RAB9AMCHR1
SCHEMBL26874763 0.82 MEN1 (0.34) MAPTMCHR1KDM4E
SCHEMBL30714683 0.82 NPC1 (0.34) NPC1RAB9AMAPTPOLBKDM4E
SCHEMBL30714690 0.82 ALOX5AP (0.40) MCHR1
SCHEMBL30714639 0.82 KDM4E (0.38) NPC1RAB9AMAPTPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-12-11 US disclosed
EP-4499624-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-02-05 EP disclosed
WO-2023230540-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS TRPV3, TRPM2, TRPV1 NPC1 349/4885RAB9A 2614/4885MAPT 2020/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.